METFORMIN HYDROCHLORIDE

METFORMIN HYDROCHLORIDE

METFORMIN HYDROCHLORIDE

Medicinal

Metformin Hydrochloride (HCl) is the active pharmaceutical ingredient (API) used in the formulation of medications for the treatment of type 2 diabetes mellitus. It belongs to the biguanide class of antidiabetic drugs.

Chemical Name: N,N-Dimethylimidodicarbonimidic diamide hydrochloride

CAS Number: 1115-70-4

Molecular Formula: C4H11N5 · HCl

Molecular Weight: 165.62 g/mol

Appearance: White to off-white crystalline powder

Solubility: Freely soluble in water, slightly soluble in alcohol

Mechanism of Action:

  • Reduces hepatic glucose production
  • Increases insulin sensitivity in peripheral tissues
  • Decreases intestinal glucose absorption

Key Features and Benefits:

  • Effective in controlling blood glucose levels in patients with type 2 diabetes.
  • Does not stimulate insulin secretion, thus minimizing the risk of hypoglycemia.
  • May have additional benefits in weight management and cardiovascular health.
  • Widely available and cost-effective API for generic drug manufacturers.

Applications:

  • Primarily used in the manufacture of oral antidiabetic tablets and extended-release formulations.
  • Combined with other antidiabetic drugs for enhanced glycemic control.

Storage and Handling:

  • Store in a tightly closed container in a cool, dry place.
  • Protect from light and moisture.
  • Handle with appropriate safety measures.

Regulatory Status:

  • Approved by major regulatory authorities for use in pharmaceutical products.
  • Subject to specific quality standards and guidelines.

Important Note:

Metformin Hydrochloride API is intended for use by pharmaceutical manufacturers and should not be consumed directly. It must be formulated into finished pharmaceutical products and administered under the supervision of a healthcare professional.

Please consult with relevant pharmaceutical regulations and guidelines for specific details and requirements for the use of Metformin Hydrochloride API in drug manufacturing.